Invention Grant
US08691807B2 Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors
有权
氮杂环丁烷基苯基,吡啶基或吡嗪基甲酰胺衍生物作为JAK抑制剂
- Patent Title: Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors
- Patent Title (中): 氮杂环丁烷基苯基,吡啶基或吡嗪基甲酰胺衍生物作为JAK抑制剂
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Application No.: US13526957Application Date: 2012-06-19
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Publication No.: US08691807B2Publication Date: 2014-04-08
- Inventor: Wenqing Yao , David M. Burns , Jincong Zhuo
- Applicant: Wenqing Yao , David M. Burns , Jincong Zhuo
- Applicant Address: US DE Wilmington
- Assignee: Incyte Corporation
- Current Assignee: Incyte Corporation
- Current Assignee Address: US DE Wilmington
- Agency: Fish & Richardson P.C.
- Main IPC: A61K31/519
- IPC: A61K31/519 ; C07D487/04

Abstract:
The present invention provides azetidinyl phenyl, pyridyl, or pyrazinyl carboxamide derivatives, as well as their compositions and methods of use, that modulate the activity of Janus kinase (JAKs) and are useful in the treatment of diseases related to the activity of JAK including, for example, inflammatory disorders, autoimmune disorders, cancer, and other diseases.
Public/Granted literature
- US20130018034A1 AZETIDINYL PHENYL, PYRIDYL OR PYRAZINYL CARBOXAMIDE DERIVATIVES AS JAK INHIBITORS Public/Granted day:2013-01-17
Information query
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