Invention Grant
US08664223B2 Pyridine and pyrimidine derivatives as inhibitors of histone deacetylase
有权
吡啶和嘧啶衍生物作为组蛋白脱乙酰酶的抑制剂
- Patent Title: Pyridine and pyrimidine derivatives as inhibitors of histone deacetylase
- Patent Title (中): 吡啶和嘧啶衍生物作为组蛋白脱乙酰酶的抑制剂
-
Application No.: US13347338Application Date: 2012-01-10
-
Publication No.: US08664223B2Publication Date: 2014-03-04
- Inventor: Laurence Françoise Bernadette Marconnet-Decrane , Sandrine Françoise Dominique Gaurrand , Patrick René Angibaud
- Applicant: Laurence Françoise Bernadette Marconnet-Decrane , Sandrine Françoise Dominique Gaurrand , Patrick René Angibaud
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica N.V
- Current Assignee: Janssen Pharmaceutica N.V
- Current Assignee Address: BE Beerse
- Agency: Baker & Hostetler LLP
- Priority: EP06100570 20060119
- Main IPC: C07D401/04
- IPC: C07D401/04 ; A61K31/444

Abstract:
This invention comprises the novel compounds of formula (I) wherein R1, R2, R3 and X have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
Public/Granted literature
- US20130143898A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE Public/Granted day:2013-06-06
Information query