Invention Grant
- Patent Title: (Aza)indole derivative substituted in position 5, pharmaceutical composition comprising it, intermediate compounds and preparation process therefor
- Patent Title (中): (Aza)吲哚衍生物,其包含其的药物组合物,中间体化合物及其制备方法
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Application No.: US12745356Application Date: 2008-12-16
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Publication No.: US08399477B2Publication Date: 2013-03-19
- Inventor: Maria Alessandra Alisi , Guido Furlotti , Nicola Cazzolla , Caterina Maugeri , Patrizia Dragone , Barbara Garofalo , Isabella Coletta , Giorgina Mangano , Beatrice Garrone
- Applicant: Maria Alessandra Alisi , Guido Furlotti , Nicola Cazzolla , Caterina Maugeri , Patrizia Dragone , Barbara Garofalo , Isabella Coletta , Giorgina Mangano , Beatrice Garrone
- Applicant Address: IT Rome
- Assignee: Aziende Chimiche Riunite Angelini Franceso A.C.R.A.F. S.p.A.
- Current Assignee: Aziende Chimiche Riunite Angelini Franceso A.C.R.A.F. S.p.A.
- Current Assignee Address: IT Rome
- Agency: Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- Priority: EP07425830 20071228
- International Application: PCT/EP2008/067622 WO 20081216
- International Announcement: WO2009/083436 WO 20090709
- Main IPC: A61K31/4439
- IPC: A61K31/4439 ; A61K31/4045 ; C07D471/04 ; C07D209/14 ; A61P35/00 ; A61P29/00 ; A61P19/02

Abstract:
An (aza)indole derivative substituted in position 5, of formula (I) in which X, Y, Z, G1, G2, G3, R1, W, and R2 have the meanings given in the description, a pharmaceutical composition comprising it, and also intermediate compounds and a preparation process therefor.
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