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US08236805B2 Substituted piperazines as CB1 antagonists 失效
取代的哌嗪作为CB1拮抗剂

Substituted piperazines as CB1 antagonists
Abstract:
Compounds of Formula (I): or pharmaceutically acceptable salts, solvates, or esters thereof, are useful in treating diseases or conditions mediated by CB1 receptors, such as metabolic syndrome and obesity, neuroinflammatory disorders, cognitive disorders and psychosis, addiction (e.g., smoking cessation), gastrointestinal disorders, and cardiovascular conditions.
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