Invention Grant
- Patent Title: Controlled release sterile injectable aripiprazole formulation and method
- Patent Title (中): 控释型无菌注射阿立哌唑制剂及方法
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Application No.: US10968482Application Date: 2004-10-19
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Publication No.: US07807680B2Publication Date: 2010-10-05
- Inventor: Janusz W. Kostanski , Takakuni Matsuda , Manoj Nerurkar , Vijay H. Naringrekar
- Applicant: Janusz W. Kostanski , Takakuni Matsuda , Manoj Nerurkar , Vijay H. Naringrekar
- Applicant Address: JP Tokyo
- Assignee: Otsuka Pharmaceutical Co., Ltd.
- Current Assignee: Otsuka Pharmaceutical Co., Ltd.
- Current Assignee Address: JP Tokyo
- Agency: Sughrue Mion, PLLC
- Main IPC: A61K31/497
- IPC: A61K31/497

Abstract:
A controlled release sterile freeze-dried aripiprazole formulation is provided which is formed of aripiprazole of a desired mean particle size and a vehicle therefor, which upon constitution with water and intramuscular injection releases aripiprazole over a period of at least about one week and up to about eight weeks. A method for preparing the controlled release freeze-dried aripiprazole formulation, and a method for treating schizophrenia employing the above formulation are also provided.
Public/Granted literature
- US20050148597A1 Controlled release sterile injectable aripiprazole formulation and method Public/Granted day:2005-07-07
Information query
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