Invention Grant
- Patent Title: Imidazoquinoline derivatives as adenosine A3 receptor ligands
- Patent Title (中): 咪唑喹啉衍生物作为腺苷A3受体配体
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Application No.: US12140512Application Date: 2008-06-17
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Publication No.: US07709489B2Publication Date: 2010-05-04
- Inventor: Peter Aranyi , Laszlo Balazs , Maria Balogh , Sandor Batori , Lajos T. Nagy , Geza Timari , Kinga Boer , Zoltan Kapui , Endre Mikus , Katalin Gerber , Judit Vargane Szeredi , Katalin Urban-Szabo , Erzsebet Walcz
- Applicant: Peter Aranyi , Laszlo Balazs , Maria Balogh , Sandor Batori , Lajos T. Nagy , Geza Timari , Kinga Boer , Zoltan Kapui , Endre Mikus , Katalin Gerber , Judit Vargane Szeredi , Katalin Urban-Szabo , Erzsebet Walcz
- Applicant Address: FR Paris
- Assignee: sanofi-aventis
- Current Assignee: sanofi-aventis
- Current Assignee Address: FR Paris
- Agent Brian R. Morrill
- Priority: HU0203976 20021115
- Main IPC: A61K31/496
- IPC: A61K31/496 ; C07D403/14 ; C07D403/06

Abstract:
This invention is directed to a compound of formula (I), wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, X, Z, m, n, o, p and r are as defined herein, its preparation, pharmaceutical composition and use as an adenosine A3 receptor ligand preferably an antagonist.
Public/Granted literature
- US20080255110A1 IMIDAZOQUINOLINE DERIVATIVES AS ADENOSINE A3 RECEPTOR LIGANDS Public/Granted day:2008-10-16
Information query
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